Home GPCR & G Protein Vasopressin Receptor Vasopressin receptor 2-Selectief Antagonists

Vasopressin receptor 2-Selectief Antagonists

  • Vasopressin receptor 1
  • Vasopressin receptor 2
Cat.nr. Productnaam Informatie Selectief / Pan IC50 / Ki
S2593 Tolvaptan Tolvaptan is an orally effective nonpeptide arginine vasopressin V2 receptor antagonist with IC50 of 3 nM, used to treat hyponatremia. Selective vasopressin receptor 2, IC50: 3 nM
S2920 Mozavaptan Mozavaptan is a novel competitive vasopressin receptor antagonist for both V1 and V2 receptors with IC50 of 1.2 μM and 14 nM, respectively. Selective Vasopressin receptor 2, IC50: 14 nM
S2116 Conivaptan HCl Conivaptan HCl is a non-peptide inhibitor of antidiuretic hormone (vasopressin receptor antagonist). Pan